Cancer Terms

Pheniramine Maleate

Cancer Terms -> Drugs and Chemicals -> Pharmacologic Substance -> Biological Response Modifier -> Histamine-1 Receptor Antagonist -> Pheniramine Maleate

Pheniramine Maleate Definition

The maleate salt form of pheniramine, an alkylamine derivative with antihistaminic and vasodilatory properties. Pheniramine maleate binds to histamine H1 receptors, thereby inhibiting phospholipase A2 and production of endothelium-derived relaxing factor, nitric oxide. Subsequent lack of activation of guanylyl cyclase through nitric oxide results in decreased cyclic GMP (cGMP) levels, thereby inhibiting constriction of smooth muscle tissue, and decreased capillary permeability and histamine-activated allergic reactions.

Pheniramine Maleate Synonyms

Pheniramine Maleate, PHENIRAMINE MALEATE

Terms in Pheniramine Maleate category



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